反応 #3973

ord-6a823073ab7c4f51901f88aec89eb947

反応方程式

CC(=O)O
acetic acid
COc1cc(C(=O)O)ccc1-c1nc2[nH]c(=O)[nH]c(=O)c2[nH]1
8-(2-methoxy-4-carboxy-phenyl)-1H,-3H-purin-2,6-dione
N
ammonia
O
water
COc1cc(C(N)=O)ccc1-c1nc2[nH]c(=O)[nH]c(=O)c2[nH]1
8-(2-Methoxy-4-aminocarbonyl-phenyl)-1H,3H-purin-2,6-dione

反応条件

詳細条件
See reaction.notes.procedure_details.

後処理

  1. 1
    その他the product precipitated
  2. 2
    ろ過is filtered off

実験手順

A quantity of 2.3 gm of 8-(2-methoxy-4-carboxy-phenyl)-1H,-3H-purin-2,6-dione are refluxed for one hour in 50 ml of thionyl chloride with the addition of 1 drop of dimethylformamide. The excess thionyl chloride is drawn off, and the residue is stirred for 16 hours at ambient temperature with a solution of ammonia in dimethylformamide. The dimethylformamide is drawn off, the remainder is mixed with water and acidified with glacial acetic acid, and the product precipitated is filtered off.

出典

DOI: 10.6084/m9.figshare.5104873.v1特許: US04722929uspto-grants-1988_02