反応 #1984

ord-593685df77934601a60a768a24ebbaa0

反応条件

詳細条件
See reaction.notes.procedure_details.

後処理

  1. 1
    その他The white precipitate was collected
  2. 2
    洗浄washed
  3. 3
    その他dried

実験手順

2-(Trifluoromethyl)acrylic acid (2.48 g, 20 mmol) was dissolved in 30 mL of dry methylene chloride, a solution of 4.75 g (20 mmol) of N-benzyl-N-(methoxymethyl)-trimethylsilylmethylamine in 20 mL of dry methylene chloride was added dropwise under N2 at 0° C. To this solution was added 2 mL of TFA, and the solution was stirred for 2 hours at room temperature. The white precipitate was collected, washed and dried to give 3.22 g of the title compound.

出典

DOI: 10.6084/m9.figshare.5104873.v1特許: US05726182uspto-grants-1998_03