4-methyl-1,3-thiazol-2-amine

Cc1csc(Nc2cccc(N3CCCOC3=O)n2)n1

収率 44.0%750 AstraZeneca ELN dataset

Cc1csc(Nc2cccc(N3CCCOC3=O)n2)n1

収率 57.2%750 AstraZeneca ELN dataset

Cc1csc(Nc2cccc(C(=O)O)n2)n1

収率 0.0%750 AstraZeneca ELN dataset

Cc1csc(Nc2cccc(N3CCOCC3=O)n2)n1

収率 80.0%750 AstraZeneca ELN dataset

Cc1csc(Nc2cccc(N3CCOCC3=O)n2)n1

収率 66.6%750 AstraZeneca ELN dataset

Cc1csc2nc(C(C)Br)cc(=O)n12

Reaction #86513

desired product

収率 42.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_09

Cc1csc(NC(=O)c2cc(Oc3ccc(-c4nnc(C)o4)cc3)cc(OC3CCN(C)C3=O)c2)n1

Reaction #163151

titled compound

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09

Br.COCCn1c(C)csc1=N

Reaction #165580

収率 34.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09

[NH4+].[OH-]

Reaction #165649

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09

Cc1nc(N)sc1C(O)(C(F)(F)F)C(F)(F)F

Reaction #165691

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09

Cc1csc(Nc2nccc3cccnc23)n1

Reaction #185421

DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)

COc1cccc(C=Cc2nc3sccn3c2C(=O)Nc2nc(C)cs2)c1OCC(C)(C)C

Reaction #187364

DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)

Cc1csc(NC(=O)c2nc(C)cc(Br)c2C)n1

Reaction #188060

DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)

Cc1csc(NCCOc2ccc(NC(=O)c3cccc(F)c3)cc2-c2ccnn2C)n1

Reaction #209461

DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)

Cc1csc(NC(=O)C2=C(O)c3sc4ccccc4c3S(=O)(=O)N2C)n1

Reaction #215443

4-Hydroxy-2-methyl-N-(4-methyl-2-thiazolyl)-2H-[1]benzothieno[2,3-e]-1,2-thiazine-3-carboxamide-1,1-dioxide

収率 66.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1981_03

Cc1ccc2c3c(sc2c1)C(O)=C(C(=O)Nc1nc(C)cs1)N(C)S3(=O)=O

Reaction #215466

2,7-Dimethyl-4-hydroxy-N-(4-methyl-2-thiazolyl)-2H-[1] benzothieno [2,3-e]-1,2-thiazine-3-carboxamide-1,1-dioxide

収率 40.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1981_03

Cc1csc(NC(=O)C2=C(O)c3sc4cc(Cl)ccc4c3S(=O)(=O)N2C)n1

Reaction #215474

7-Chloro-4-hydroxy-2-methyl-N-(4-methyl-2-thiazolyl)-2H-[1] benzothieno [2,3-e]-1,2-thiazine-3-carboxamide-1,1-dioxide

収率 36.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1981_03

CCOC(=O)c1cnc(Nc2nc(C)cs2)cc1Oc1ccccc1

Reaction #224761

DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (9/10)

Cc1csc(NC(=O)c2cc(Oc3cnc(C(=O)N4CCC4)cn3)cc(OC3CCOC3)c2)n1

Reaction #233955

DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (9/10)

Cc1csc(NC(=O)CBr)n1

Reaction #234510

DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (9/10)

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