Réaction #70345

ord-2e7264dd618b47aeb93ca0f50ac17746

Conditions de réaction

Conditions détaillées
See reaction.notes.procedure_details.

Traitement

  1. 1
    AutreObtained
  2. 2
    Autre(0.152 g, 63% of yield)

Mode opératoire

Obtained (0.152 g, 63% of yield) following the procedure described in Example 14 (step C) starting with tert-butyl 2-(6-(2-chlorophenyl)-5-methylpyridin-3-ylamino)-5-methylbenzoate (0.49 mmol, 0.200 g) and cyclopropylboronic acid (1.47 mmol, 0.126 g).

Source

DOI: 10.6084/m9.figshare.5104873.v1Brevet: US08536165B2uspto-grants-2013_09