Reacción #81660

ord-43c2d0092e9e45ee9a564bd57c4bb551

Ecuación de reacción

CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(C)(C)CCC3=O)cc1
ethyl 4-[(5,6,7,8-tetrahydro-8,8-dimethyl-5-oxonaphth-2-yl)ethynyl]benzoate
CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(C)(C)CCC3=O)cc1
Compound 1
CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(C)(C)CCC3=O)cc1
ethyl 4-[(5,6,7,8-tetrahydro-8,8-dimethyl-5-oxonaphth-2-yl)ethynyl]benzoate
C#Cc1ccc2c(c1)C(=O)CCC2(C)C
7-ethynyl-3,4-dihydro-4,4-dimethylnaphthalen-1(2H)-one
C#Cc1ccc2c(c1)C(=O)CCC2(C)C
Compound L
C#Cc1ccc2c(c1)C(=O)CCC2(C)C
7-ethynyl-3,4-dihydro-4,4-dimethylnaphthalen-1(2H)-one
CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(=O)CCC3(C)C)cc1
title compound
CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(=O)CCC3(C)C)cc1
Ethyl 4-[(5,6,7,8-tetrahydro-8,8-dimethyl-5-oxonaphth-3-yl)ethynyl]benzoate

Condiciones de reacción

Condiciones detalladas
See reaction.notes.procedure_details.

Procedimiento

Employing the same general procedure as for the preparation of ethyl 4-[(5,6,7,8-tetrahydro-8,8-dimethyl-5-oxonaphth-2-yl)ethynyl]benzoate (Compound 1), 4 g (21.7 mmol ) of 7-ethynyl-3,4-dihydro-4,4-dimethylnaphthalen-1(2H)-one (Compound L) was converted into the title compound using 6 g (21.7 mmol) of ethyl 4-iodobenzoate, 5 g (7.2 mmol) of bis(triphenylphosphine)palladium(II) chloride and 1.4 g (7.2 mmol) of cuprous iodide.

Fuente

DOI: 10.6084/m9.figshare.5104873.v1Patente: US05618931uspto-grants-1997_04