Reacción #70896

ord-b2f46e59caa549ac85c950c66cafc547

Condiciones de reacción

Condiciones detalladas
See reaction.notes.procedure_details.

Procedimiento

Following a similar procedure to that described in example 48, but starting from 2-(2-aminoethyl)-4,6-bis(4-fluorophenyl)-5-(4-pyridyl)pyrazolo[3,4-b]pyridine (obtained in example 90) and 1-(tert-butoxycarbonyl)piperidine-4-carboxylic acid, the desired compound was obtained.

Fuente

DOI: 10.6084/m9.figshare.5104873.v1Patente: US08536194B2uspto-grants-2013_09