Reacción #60179

ord-a8faa2e9ef8449eaa429ddd5da92288b

Ecuación de reacción

COc1cc(Cl)ccc1C(=O)Cl
4-chloro-2-methoxybenzoyl chloride
N#Cc1ccc(Cl)nc1
2-chloro-5-(cyano)pyridine
O=[N+]([O-])c1ccc(NCCNc2ncc(-c3ncc[nH]3)c(-c3ccc(Cl)cc3Cl)n2)nc1
[4-(2,4-dichlorophenyl)-5-imidazol-2-ylpyrimidin-2-yl]{2-[(5-nitro(2-pyridyl))amino]ethyl}amine
COc1cc(Cl)ccc1-c1nc(NCCNc2ccc(C#N)cn2)ncc1-c1ncc[nH]1
6-[(2-{[4-(4-chloro-2-methoxyphenyl)-5-imidazol-2-ylpyrimidin-2-yl]amino}-ethyl)amino]pyridine-3-carbonitrile

Condiciones de reacción

Condiciones detalladas
See reaction.notes.procedure_details.

Procedimiento

6-[(2-{[4-(4-chloro-2-methoxyphenyl)-5-imidazol-2-ylpyrimidin-2-yl]amino}-ethyl)amino]pyridine-3-carbonitrile was prepared from 4-chloro-2-methoxybenzoyl chloride and 2-chloro-5-(cyano)pyridine using the general method for [4-(2,4-dichlorophenyl)-5-imidazol-2-ylpyrimidin-2-yl]{2-[(5-nitro(2-pyridyl))amino]ethyl}amine.

Fuente

DOI: 10.6084/m9.figshare.5104873.v1Patente: US07425557B2uspto-grants-2008_09