Reacción #572088

ord-a18fc874d8fc41589f82a55438ee021e

Condiciones de reacción

Condiciones detalladas
See reaction.notes.procedure_details.

Procedimiento

The same procedures for preparing 1-(3-diethylaminopropyl)-3-amino-4-chloroindazole as described in Example 89 were repeated except that 8 g of 3-phthalimidoindazole and 9.5 g of 3-bromopropylpyrrolidine hydrobromide were employed instead of the 3-phthalimido-4-chloroindazole and the 3-bromopropyldiethylamine hydrobromide, respectively. As a result, 8.2 g of 1-(3-pyrrolidinopropyl)-3-aminoindazole was obtained.

Fuente

DOI: 10.6084/m9.figshare.5104873.v1Patente: US04533731uspto-grants-1985_08