Reacción #433848

ord-a739cdb553fe4e229ecd8ac9f8217cf9

Condiciones de reacción

Condiciones detalladas
See reaction.notes.procedure_details.

Procedimiento

Using an analogous procedure to that described in Example 4, 4-[1-(4-pyridyl)piperidin-4-yloxy]aniline was reacted with 4-toluenesulphonyl chloride to give N-{4-[1-(4-pyridyl)piperidin-4-yloxy]phenyl}-4-toluenesulphonamide, hydrochloride salt, in 54% yield, m.p. 270-272° C.;

Fuente

DOI: 10.6084/m9.figshare.5104873.v1Patente: US07173025B1uspto-grants-2007_02