Reacción #2329554

Ecuación de reacción

5-cyano-1-(3-trifluoromethoxybenzyl)-1H-indole-2-carboxylic acid

2-amino-2-(tetrahydropyran-4-yl)ethanol

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title compound

5-Cyano-1-(3-trifluoromethoxybenzyl)-1H-indole-2-carboxylic acid [2-hydroxy-1-(tetrahydropyran-4-yl)ethyl]amide

Condiciones de reacción

Procedimiento

The title compound was prepared using 5-cyano-1-(3-trifluoromethoxybenzyl)-1H-indole-2-carboxylic acid [prepared from 3-(trifluoromethoxy)benzyl bromide and ethyl 5-cyanoindole-2-carboxylate] and 2-amino-2-(tetrahydropyran-4-yl)ethanol in a manner similar to that described in Example 11.

Fuente