Reacción #2074998

ord-50f4a76b35d54c17ba67c92dcef22690

Ecuación de reacción

O=C(Cl)c1ccc2cc(Br)ccc2c1
6-Bromo-naphthalene-2-carbonyl chloride
Nc1ccc2[nH]cnc2c1
1H-benzoimidazol-5-ylamine
O=C(Nc1ccc2[nH]cnc2c1)c1ccc2cc(Br)ccc2c1
title compound
O=C(Nc1ccc2[nH]cnc2c1)c1ccc2cc(Br)ccc2c1
6-Bromo-naphthalene-2-carboxylic acid (1H-benzoimidazol-5-yl)-amide

Condiciones de reacción

Condiciones detalladas
See reaction.notes.procedure_details.

Tratamiento posterior

  1. 1
    OtroThis material was prepared analogous to the procedure

Procedimiento

This material was prepared analogous to the procedure described for Example 1 (b). 6-Bromo-naphthalene-2-carbonyl chloride, Example 1(a), reacted with 1H-benzoimidazol-5-ylamine (TimTec) to give the title compound as an amorphous solid. MS (ESI, pos. ion.) m/z: 366 (M+1).

Fuente

DOI: 10.6084/m9.figshare.5104873.v1Patente: US07553848B2uspto-grants-2009_06