Reacción #11046

ord-d92c58b0faca44eeb43c64c494c5501b

Ecuación de reacción

CCOC(=O)CC(NS(=O)(=O)c1cccc(-c2cccc(Nc3nccs3)c2)c1)c1ccccc1
Ethyl 3-phenyl-3-{[3′-(1,3-thiazol-2-ylamino)[1,1′-biphenyl]-3-yl]sulfonylamino}-propanoate
CCOC(C)=O.ClCCl
dichloromethane methanol
CCOC(C)=O.ClCCl
dichloromethane acetic acid ethyl ester
O=C(O)CC(NS(=O)(=O)c1cccc(-c2cccc(Nc3nccs3)c2)c1)c1ccccc1
3-phenyl-3-{[3′-(1,3-thiazol-2-ylamino)[1,1′-biphenyl]-3-yl]sulfonylamino}-propanoic acid

Condiciones de reacción

Condiciones detalladas
See reaction.notes.procedure_details.

Procedimiento

0.2 g of Ethyl 3-phenyl-3-{[3′-(1,3-thiazol-2-ylamino)[1,1′-biphenyl]-3-yl]sulfonylamino}-propanoate 15.1.1 were saponified in 15 ml dimethoxyethane 12 ml water and 0.2 g LiOH. After aqueos work-up and flash chromatography (dichloromethane/methanol 10+1) 65 mg were obtained.

Fuente

DOI: 10.6084/m9.figshare.5104873.v1Patente: US07094911B2uspto-grants-2006_08