Reaction #690465

ord-7cfd7e423b0b41ee84b4c03f548be02d

Reaction equation

CC(=O)Oc1ccc2c(c1)OCC(c1ccccc1)=C2
7-acetoxyisoflav-3-ene
c1c[nH]cn1
imidazole
Oc1ccc(C2=Cc3ccc(O)cc3OC2)cc1
isoflav-3-ene-4′,7-diol
Oc1ccc2c(c1)OCC(c1ccccc1)=C2
Isoflav-3-ene-7-ol

Solvents

Conditions

Detailed conditions
See reaction.notes.procedure_details.

Procedure

Isoflav-3-ene-7-ol was prepared from 7-acetoxyisoflav-3-ene (0.2 g, 0.75 mmol) and imidazole (0.24 g) in ethanol (3.5 ml) as described for isoflav-3-ene-4′,7-diol. Yield: (0.11 g, 66%) m.p. 120° C. 1H NMR (d6-DMSO): δ 5.07 (s, 2H, H2), 6.24 (d, 1H, J 2.2 Hz, H8), 6.33 (dd, 1H, J 1.9 Hz, 7.9 Hz, H6), 6.96 (d, 1H, J 7.9 Hz, H5), 7.00 (s, 1H, H4), 7.26-7.47 (m, 5H, ArH), 9.65 (bs, 1H, OH). Mass spectrum: m/z 224 (m, 74%); 223 (100), 175 (28); 165 (23); 147 (41).

Source

DOI: 10.6084/m9.figshare.5104873.v1Patent: US07906660B2uspto-grants-2011_03