Reaction #1147643
ord-160c4de64cc04cfd9a8834898fc652bb
Reaction equation
2,6-Dimethoxy-3-(hydroxymethyl)benzeneboronic acid
N-(2,6-dichlorobenzoyl)-4-bromo-L-phenylalanine ethyl ester
→
N-(2,6-dichlorobenzoyl)-4-[2,6-dimethoxy-3-(hydroxymethyl)phenyl]-L-phenylalanine ethyl ester
Reactants
Reagents
None
Conditions
Detailed conditions
See reaction.notes.procedure_details.
Procedure
2,6-Dimethoxy-3-(hydroxymethyl)benzeneboronic acid was coupled with N-(2,6-dichlorobenzoyl)-4-bromo-L-phenylalanine ethyl ester in a similar method as described in Example 7-2) to give N-(2,6-dichlorobenzoyl)-4-[2,6-dimethoxy-3-(hydroxymethyl)phenyl]-L-phenylalanine ethyl ester.