Reaction #1139712

ord-952593db26c4400b81b43c652b55dcbc

Conditions

Detailed conditions
See reaction.notes.procedure_details.

Procedure

6-Bromo-1H-indazole (500 mg, 2.54 mmol) was treated with 4-methoxybenzene-1-sulfonyl chloride (576 mg, 2.79 mmol) according to the method described in Preparation 15b to give 820 mg (81% yield) of the title compound. Purity 92%.

Source

DOI: 10.6084/m9.figshare.5104873.v1Patent: US09388189B2uspto-grants-2016_07