Reaction #1006026

ord-abd02e89de774ad0af8caf0d39fce101

Reaction equation

NCc1ccc2c(c1)OCCCO2
(3,4-dihydro-2H-benzo[b][1,4]dioxepin-7-yl)methanamine
CCOC(=O)c1cn2cc(Br)ccc2n1
ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate
O=C(NCc1ccc2c(c1)OCCCO2)c1cn2cc(Br)ccc2n1
title compound
O=C(NCc1ccc2c(c1)OCCCO2)c1cn2cc(Br)ccc2n1
6-Bromo-N-((3,4-dihydro-2H-benzo[b][1,4]dioxepin-7-yl)methyl)imidazo[1,2-a]pyridine-2-carboxamide

Conditions

Detailed conditions
See reaction.notes.procedure_details.

Procedure

The title compound was prepared by essentially following the same procedures described for Intermediate I, using (3,4-dihydro-2H-benzo[b][1,4]dioxepin-7-yl)methanamine and ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate as starting materials.

Source

DOI: 10.6084/m9.figshare.5104873.v1Patent: US09271969B2uspto-grants-2016_03