Reaction #1006024

ord-1d20ba7682d24bb6b50bd8b1ed0de881

Reaction equation

COc1ccc(CN)cc1OC
(3,4-dimethoxyphenyl)methanamine
CCOC(=O)c1cn2cc(Br)ccc2n1
ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate
COc1ccc(CNC(=O)c2cn3cc(Br)ccc3n2)cc1OC
title compound
COc1ccc(CNC(=O)c2cn3cc(Br)ccc3n2)cc1OC
6-Bromo-N-(3,4-dimethoxybenzyl)imidazo[1,2-a]pyridine-2-carboxamide

Conditions

Detailed conditions
See reaction.notes.procedure_details.

Procedure

The title compound was prepared by essentially following the same procedures described for Intermediate I, using (3,4-dimethoxyphenyl)methanamine and ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate as starting materials.

Source

DOI: 10.6084/m9.figshare.5104873.v1Patent: US09271969B2uspto-grants-2016_03