Reaction #1006020

ord-c9d35595ea1f4502ab0988e53e80beb1

Reaction equation

CC(C)c1ccc(CN)cc1
(4-isopropylphenyl)methanamine
CCOC(=O)c1cn2cc(Br)ccc2n1
ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate
CC(C)c1ccc(CNC(=O)c2cn3cc(Br)ccc3n2)cc1
title compound
CC(C)c1ccc(CNC(=O)c2cn3cc(Br)ccc3n2)cc1
6-Bromo-N-(4-isopropylbenzyl)imidazo[1,2-a]pyridine-2-carboxamide

Conditions

Detailed conditions
See reaction.notes.procedure_details.

Procedure

The title compound was prepared by essentially following the same procedures described for Intermediate I, using (4-isopropylphenyl)methanamine and ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate as starting materials.

Source

DOI: 10.6084/m9.figshare.5104873.v1Patent: US09271969B2uspto-grants-2016_03