Reaction #1006015

ord-3a0f2042c7774c0aa4c665fdd58d0018

Reaction equation

NCc1ccc2c(c1)OCO2
benzo[d][1,3]dioxol-5-ylmethanamine
CCOC(=O)c1cn2cc(Br)ccc2n1
ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate
O=C(NCc1ccc2c(c1)OCO2)c1cn2cc(Br)ccc2n1
title compound
O=C(NCc1ccc2c(c1)OCO2)c1cn2cc(Br)ccc2n1
N-(Benzo[d][1,3]dioxol-5-ylmethyl)-6-bromoimidazo[1,2-a]pyridine-2-carboxamide

Conditions

Detailed conditions
See reaction.notes.procedure_details.

Procedure

The title compound was prepared by essentially following the same procedures described for Intermediate I, using benzo[d][1,3]dioxol-5-ylmethanamine and ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate as starting materials.

Source

DOI: 10.6084/m9.figshare.5104873.v1Patent: US09271969B2uspto-grants-2016_03