Reaction #1006004

ord-6f3836246ec94f7d89de56932a4618e3

Reaction equation

Nc1ccc(OC(F)(F)F)cc1
4-(trifluoromethoxy)aniline
CCOC(=O)c1cn2cc(Br)ccc2n1
ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate
O=C(Nc1ccc(OC(F)(F)F)cc1)c1cn2cc(Br)ccc2n1
title compound
O=C(Nc1ccc(OC(F)(F)F)cc1)c1cn2cc(Br)ccc2n1
6-Bromo-N-(4-(trifluoromethoxy)phenyl)imidazo[1,2-a]pyridine-2-carboxamide

Conditions

Detailed conditions
See reaction.notes.procedure_details.

Procedure

The title compound was prepared by essentially following the same procedures described for Intermediate I, using 4-(trifluoromethoxy)aniline and ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate as starting materials.

Source

DOI: 10.6084/m9.figshare.5104873.v1Patent: US09271969B2uspto-grants-2016_03