(S)-3-(3-(tert-butyldimethylsilyl-oxy)azetidin-1-yl)-2-hydroxy-N-(5-methylpyrazin-2-yl)propanamide

Cc1cnc(NC(=O)[C@H](CN2CC(O[Si](C)(C)C(C)(C)C)C2)Oc2ncnc3c2cnn3-c2c(Cl)cccc2Cl)cn1
Reaction #742299
product
Yield 57.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_12
Cc1cnc(NC(=O)[C@H](CN2CC(O[Si](C)(C)C(C)(C)C)C2)Oc2ncnc3c2cnn3-c2ccccc2Cl)cn1
Reaction #1185447
product
Yield 82.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2012_03
Cc1cnc(NC(=O)[C@H](CN2CC(O[Si](C)(C)C(C)(C)C)C2)Oc2ncnc3c2cnn3-c2c(Cl)cccc2Cl)cn1
Reaction #1185449
product
Yield 57.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2012_03