HATU

NCC(F)(F)CNC(=O)c1ccc(F)c(NCc2cnc(Nc3ccccn3)s2)c1
Reaction #6980
title compound
Yield 65.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2006_08
C#CC(=O)NC1CCCN(C(=O)[C@H](C)N2CC[C@H](NS(=O)(=O)c3ccc4cc(Cl)ccc4c3)C2=O)C1
Reaction #7399
title compound
Yield 115.5%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2006_08
CCN(CC)CCNC(=O)c1ccc2[nH]c(-c3cc(-c4ccncc4)n[nH]c3=O)nc2c1
Reaction #40544
2-(3-Oxo-6-pyridin-4-yl-2,3-dihydropyridazin-4-yl)-1H-benzimidazole-5-carboxylic acid (2-diethylaminoethyl)amide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
O=C(/C=C/c1ccc(-c2ccc(O)c(Cl)c2)cc1)NO
Reaction #41267
title compound
Yield 9.7%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Cc1nnc(C(=O)N[C@@H](C)[C@H](Oc2ccc3c(cnn3-c3ccc(F)cc3)c2)c2ccccc2)o1
Reaction #41420
N-{(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl}-5-methyl-[1,3,4]oxadiazol-2-carboxamide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
C[C@H](NC(=O)C1(C)CC1)[C@H](Oc1ccc2c(cnn2-c2ccc(F)cc2)c1)c1ccc2c(c1)OCCO2
Reaction #41431
N-((1R,2S)-1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1-(1-(4-fluorophenyl)-1H-indazol-5-yloxy)propan-2-yl)-1-methylcyclopropanecarboxamide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
C[C@H](NC(=O)[C@@H]1CCCN1)[C@H](Oc1ccc2c(cnn2-c2ccc(F)cc2)c1)c1ccc2c(c1)OCCO2
Reaction #41432
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COc1cccc([C@@H](Oc2ccc3c(cnn3-c3ccc(Cl)cc3)c2)[C@H](C)NC(=O)C(C)(F)F)c1
Reaction #41435
crude product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Cc1cnc(C(=O)N[C@@H](C)[C@H](Oc2ccc3c(cnn3-c3ccc(F)cc3)c2)c2ccc(C)c(C)c2)s1
Reaction #41467
N-[(1R,2S)-1-(3,4-dimethylphenyl)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-propan-2-yl]-5-methyl-1,3-thiazole-2-carboxamide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
O=Cc1ccc(C(=O)NCCN2CCC(OC(=O)Nc3ccccc3-c3ccccc3)CC2)cc1
Reaction #42134
title intermediate
Yield 92.2%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
NCc1ccc(NC(=O)CCN2CCC(OC(=O)Nc3ccccc3-c3ccccc3)CC2)cc1
Reaction #42138
title intermediate
Yield 94.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
O=Cc1ccc(NC(=O)CCN2CCC(OC(=O)Nc3ccccc3-c3ccccc3)CC2)cc1
Reaction #42139
title intermediate
Yield 66.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCCNC(=O)c1cc(C(=O)N(CCC)[C@@H](Cc2ccccc2)[C@H](O)CNCc2cccc(OC)c2)cc(S(N)(=O)=O)c1
Reaction #42294
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCCN(CCC)C(=O)c1cc(CC#N)cc(C(=O)N[C@@H](Cc2ccccc2)[C@H](O)CNCc2cccc(OC)c2)c1
Reaction #42303
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCCN(CCC)C(=O)c1cc(C(=O)N[C@@H](Cc2cc(F)cc(F)c2)[C@H](O)CNCc2cccc(CC)c2)cc(-c2noc(C)n2)c1.Cl
Reaction #42339
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCCN(C)C(=O)c1cc(I)cc(C(=O)OC)c1
Reaction #42343
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCCN(C)C(=O)c1cc(C(=O)N[C@@H](Cc2ccccc2)[C@H](O)CNCc2cccc(CC)c2)cc(-c2ncco2)c1
Reaction #42345
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCc1cccc(CNC[C@@H](O)[C@H](Cc2cc(F)cc(F)c2)NC(=O)c2cccc(C(=O)OC)c2)c1
Reaction #42354
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COC(=O)c1cccc(C(=O)NC(CO)CCOCc2ccccc2)c1
Reaction #42358
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCc1cccc(CNC[C@@H](O)[C@H](Cc2cc(F)cc(F)c2)NC(=O)c2cccc(-c3nc(CCO)co3)c2)c1
Reaction #42359
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Page 1Next