Reaktion #94583

ord-3344caeaf82c468584f2bd9f26954ca1

Reaktionsgleichung

NC1CCN(CCc2c[nH]c3ccccc23)CC1.O
3-[2-(4-amino-1-piperidyl)ethyl]indole monohydrate
O=S(=O)(Cl)C1CCCCC1
cyclohexanesulphonyl chloride
→
O=S(=O)(NC1CCN(CCc2c[nH]c3ccccc23)CC1)C1CCCCC1
title compound
O=S(=O)(NC1CCN(CCc2c[nH]c3ccccc23)CC1)C1CCCCC1
3-[2-(4-Cyclohexanesulphonamido-1-piperidyl)ethyl]indole

Edukte

NC1CCN(CCc2c[nH]c3ccccc23)CC1.O
3-[2-(4-amino-1-piperidyl)ethyl]indole monohydrate
O=S(=O)(Cl)C1CCCCC1
cyclohexanesulphonyl chloride

Reagenzien

Keine

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

Using an analogous procedure to Example 1 3-[2-(4-amino-1-piperidyl)ethyl]indole monohydrate may be reacted with cyclohexanesulphonyl chloride to give the title compound.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US04131680uspto-grants-1978_12