Reaktion #94059

ord-1b0a258bfe104ae1a025a9460502811f

Reaktionsgleichung

CCCCN=C1c2ccccc2CCc2c1nc1c(cnn1CC)c2NCCCC
N-butyl-11-(butylimino)-1-ethyl-1,5,6,11-tetrahydrobenzo[5,6]cyclohepta[1,2-b]pyrazolo[4,3-e]pyridin-4-amine
O=S(=O)(O)O
sulfuric acid
CCCCNc1c2c(nc3c1cnn3CC)C(=O)c1ccccc1CC2
4-(Butylamino)-1-ethyl-5,6-dihydrobenzo[5,6]cyclohepta[1,2-b]pyrazolo[4,3-e]pyridin-11(1H)-one

Lösungsmittel

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

7.2 g. of N-butyl-11-(butylimino)-1-ethyl-1,5,6,11-tetrahydrobenzo[5,6]cyclohepta[1,2-b]pyrazolo[4,3-e]pyridin-4-amine (0.018 mol.) and 100 ml. of aqueous sulfuric acid (30%) are reacted according to the procedure of Example 6, yield: 4.7 g. (75%); m.p. 181°-183° (ethyl acetate/ether).

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US04128717uspto-grants-1978_12