Reaktion #81448

ord-54b4091bbb124d768a7411fc5e06240b

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Aufarbeitung

  1. 1
    SonstigeThe yield obtained

Vorschrift

The method of operation is the same as that used for the synthesis of the compound of Example 1 (coupling with 1-ethoxy-1-(trimethylstannyl)ethylene), 2-benzyloxy-6-bromooxazolo[4,5-b]pyridine from Preparation 4 being used instead of the 6-bromo-3-methyloxazolo[4,5-b]pyridin-2(3H)-one from Preparation 2. The yield obtained is 78%. ##STR49##

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US05618819uspto-grants-1997_04