Reaktion #78976

ord-b1cd9084cdec4146813e37bf30419a1c

Reaktionsgleichung

Nc1ccc(-c2cccc(Cl)c2)cc1C(=O)C1CC1
(4-amino-3′-chloro-biphenyl-3-yl)-cyclopropyl-methanone
[Br][Mg][CH]1CC1
cyclopropylmagnesium bromide
Nc1ccc(-c2cccc(Cl)c2)cc1C(O)(C1CC1)C1CC1
(4-Amino-3′-chloro-biphenyl-3-yl)-dicyclopropyl-methanol

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

(4-Amino-3′-chloro-biphenyl-3-yl)-dicyclopropyl-methanol (mp 90-92° C.; MS ((+)ESI) m/z 314 (M+H)+.) was prepared from (4-amino-3′-chloro-biphenyl-3-yl)-cyclopropyl-methanone and cyclopropylmagnesium bromide according to Example 41.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US06713478B2uspto-grants-2004_03