Reaktion #7661

Reaktionsgleichung

6-(1-aminopropyl)-3-cyclopentyl-1,2,4-triazin-5(4H)-one

1-[(benzyloxy)carbonyl]-4-piperidinecarboxylic acid

→

Benzyl 4-({[1-(3-cyclopentyl-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl)propyl]amino}carbonyl)-1-piperidinecarboxylate

Reaktionsbedingungen

Aufarbeitung

1. 1
   SonstigeThe crude product is used in the next step without further purification

Vorschrift

In analogy to the procedure for Example 58A, 300 mg (1.35 mmol) 6-(1-aminopropyl)-3-cyclopentyl-1,2,4-triazin-5(4H)-one, 355 mg (1.35 mmol) 1-[(benzyloxy)carbonyl]-4-piperidinecarboxylic acid and proportionate amounts of the other reagents are used. The crude product is used in the next step without further purification.

Quelle