Reaktion #60886

ord-e234f51f109e4e5eaf0019c229d972c1

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

The title compound was prepared by a similar process to that described for Example 8 but using 6-(4-iodo-1-methyl-1H-imidazol-5-yl)-4-(methylsulfonyl)thieno[2,3-d]pyrimidine (Intermediate 94) in place of 6-(1-methyl-4-phenyl-1H-imidazol-5-yl)-4-(methylsulfonyl)thieno[2,3-d]pyrimidine (intermediate 17). Beige solid (143 mg, 85%);

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US07427616B2uspto-grants-2008_09