Reaktion #539841

Reaktionsgleichung

(1S)-1-[5-(3-bromo-1-benzofuran-5-yl)-1,3,4-oxadiazol-2-yl]ethyl acetate

(2-chloro-5-fluorophenyl)boronic acid

→

title compound

Ausbeute 66.0%

(1S)-1-[5-[3-(2-chloro-5-fluorophenyl)-1-benzofuran-5-yl]-1,3,4-oxadiazol-2-yl]ethyl acetate

Ausbeute 66.0%

Reaktionsbedingungen

Vorschrift

In the same manner as in Reference Example 19 and using (1S)-1-[5-(3-bromo-1-benzofuran-5-yl)-1,3,4-oxadiazol-2-yl]ethyl acetate instead of methyl 3-iodoimidazo[1,2-a]pyridine-6-carboxylate and (2-chloro-5-fluorophenyl)boronic acid instead of (4-methoxyphenyl)boronic acid, the title compound (yield 66%) was obtained as colorless crystals.

Quelle