Reaktion #52967

Reaktionsgleichung

2,6-Dimethoxy-3-(hydroxymethyl)benzeneboronic acid

N-(2,6-dichlorobenzoyl)-4-bromo-L-phenylalanine ethyl ester

→

N-(2,6-dichlorobenzoyl)-4-[2,6-dimethoxy-3-(hydroxymethyl)phenyl]-L-phenylalanine ethyl ester

Reaktionsbedingungen

Vorschrift

2,6-Dimethoxy-3-(hydroxymethyl)benzeneboronic acid was coupled with N-(2,6-dichlorobenzoyl)-4-bromo-L-phenylalanine ethyl ester in a similar method as described in Example 7-2) to give N-(2,6-dichlorobenzoyl)-4-[2,6-dimethoxy-3-(hydroxymethyl)phenyl]-L-phenylalanine ethyl ester.

Quelle