Reaktion #464692

ord-3212f7b590b4430483b6c6024c3e6bfd

Reaktionsgleichung

CCc1ncc[nH]1
2-ethylimidazole
C1=CCCCC1
cyclohexene
O=C(n1ccnc1)n1ccnc1
carbonyidiimidazole
O=[N+]([O-])c1c(Cl)ncnc1Cl
4,6-dichloro-5-nitropyrimidine
CNC1CCN(C)CC1
1-methyl-4-(methylamino)piperidine
CCc1ncc2c(=O)[nH]c3c(NCC4CCN(C)CC4)ncnc3n12
9-Ethyl-4-[(1-methylpiperidin-4-yl)methylamino]imidazo[5,1 -h]pteridin-6(5H)-one

Lösungsmittel

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

Prepared by treatment of 4,6-dichloro-5-nitropyrimidine with 1-methyl-4-(methylamino)piperidine followed by reaction with 2-ethylimidazole, reduction with palladium on carbon and cyclohexene in refluxing ethanol, and cyclization with carbonyidiimidazole.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US06025489uspto-grants-2000_02