Reaktion #446530

ord-e914668a7438475a80d2827f7442899a

Reaktionsgleichung

CC(C)[C@H](N)CO
valinol
O=C(Cl)CCl
chloroacetyl chloride
CC(C)C1COCC(=O)N1
5-(2-propyl)-3-morpholinone

Reagenzien

Keine

Lösungsmittel

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

Treatment of valinol in basic ethanol with chloroacetyl chloride using the procedure of Surry, et. al., J. Am. Chem. Soc. (1955) 77, 633, gives 5-(2-propyl)-3-morpholinone. Deprotonation of the latter with NaH in DMF solution and reaction with methyl iodide gives the title compound.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US05001113uspto-grants-1991_03