Reaktion #44085

ord-4c593e3f20c1418791a9340ba3606ca7

Reaktionsgleichung

Cc1ccc2c(N3CCN(CCc4cccc(N)c4)CC3)cccc2n1
3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}aniline
Cc1ccc2c(N3CCN(CCc4cccc(N)c4)CC3)cccc2n1
3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}aniline
CCCS(=O)(=O)Cl
propanesulfonyl chloride
CCCS(=O)(=O)Nc1cccc(CCN2CCN(c3cccc4nc(C)ccc34)CC2)c1
title compound
Ausbeute 62.0%
CCCS(=O)(=O)Nc1cccc(CCN2CCN(c3cccc4nc(C)ccc34)CC2)c1
N-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-1-propanesulfonamide
Ausbeute 62.0%

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

The title compound was prepared in 62% yield using a similar procedure to example E43 starting from 3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}aniline (D6) and propanesulfonyl chloride.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US07732600B2uspto-grants-2010_06