Reaktion #43116

ord-1a26662e7b0f40a1998da26103818dae

Reaktionsgleichung

O=Cc1cccc(-c2ccnc(Cl)n2)c1
Intermediate 1
O=Cc1cccc(-c2ccnc(Cl)n2)c1
3-(2-Chloro-pyrimidin-4-yl)-benzaldehyde
Nc1cccnc1
3-aminopyridine
Clc1nccc(-c2cccc(CNc3cccnc3)c2)n1
[3-(2-Chloro-pyrimidin-4-yl)-benzyl]-pyridin-3-yl-amine

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

Intermediate 1 was coupled with 3-aminopyridine following procedure B. LC-MS showed the product had the expected M+H+ of 297.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US07732444B2uspto-grants-2010_06