Reaktion #352943

ord-f0f81bb389e747fb984060e82ca15e3c

Reaktionsgleichung

CCOC(=O)CCCc1ccc(Br)cc1
ethyl 4-(4-bromophenyl)butanoate
CCOC(=O)Cc1cccc(Br)c1
ethyl (3-bromophenyl)acetate
CCOC(=O)Cc1cccc(Br)c1
ethyl 3-bromophenylacetate
CCOC(=O)Cc1cccc(Br)c1
Compound B
CCOC(=O)Cc1cccc(Br)c1
ethyl 3-bromophenylacetate
CCOC(=O)CCCc1cccc(Br)c1
title compound
CCOC(=O)CCCc1cccc(Br)c1
Ethyl 4-(3-bromophenyl)butanoate

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

Employing the same general multistep preparation as for ethyl 4-(4-bromophenyl)butanoate (Compound 60 g (246 mmol) of ethyl (3-bromophenyl)acetate (Compound B) was converted into the title compound (oil) using 255 ml (255 mmol) of diisobutylaluminum hydride (DIBAL-H, 1M in hexane), 85.8 g (250 mmol) of (carbethoxymethylene)triphenylphosphorane and 1.7 g of 10% Pd/C.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US05648514uspto-grants-1997_07