Reaktion #1946108

Reaktionsgleichung

1-(tert-butoxycarbonyl)-3-ethyl-hexahydro-1H-1,4-diazepine

5-chlorosulfonyl-4-methylisoquinoline

→

objective compound

Ausbeute 34.5%

2-Ethyl-hexahydro-1-[(4-methyl-5-isoquinolinyl)sulfonyl]-1H-1,4-diazepine hydrochloride

Ausbeute 34.5%

Reaktionsbedingungen

Vorschrift

Using 0.68 g of 1-(tert-butoxycarbonyl)-3-ethyl-hexahydro-1H-1,4-diazepine and 0.72 g of 5-chlorosulfonyl-4-methylisoquinoline, the procedure of Example 1 was otherwise repeated to provide 0.38 g of the objective compound (white crystals).

Quelle