Reaktion #1731086

ord-e609acf8a9f54153804ea4129ce7377d

Reaktionsgleichung

O=S(=O)(NC1CNc2ccc(Br)cc2C1)c1ccccc1
87A
O=S(=O)(NC1CNc2ccc(Br)cc2C1)c1ccccc1
N-(6-Bromo-1,2,3,4-tetrahydroquinolin-3-yl)-benzenesulfonamide
OB(O)c1ccccc1
phenylboronic acid
→
O=S(=O)(NC1CNc2ccc(-c3ccccc3)cc2C1)c1ccccc1
Compound 170A
O=S(=O)(NC1CNc2ccc(-c3ccccc3)cc2C1)c1ccccc1
N-(6-Phenyl-1,2,3,4-tetrahydroquinolin-3-yl)benzenesulfonamide

Edukte

O=S(=O)(NC1CNc2ccc(Br)cc2C1)c1ccccc1
87A
O=S(=O)(NC1CNc2ccc(Br)cc2C1)c1ccccc1
N-(6-Bromo-1,2,3,4-tetrahydroquinolin-3-yl)-benzenesulfonamide
OB(O)c1ccccc1
phenylboronic acid

Reagenzien

Keine

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

Compound 170A was prepared from 87A and phenylboronic acid by procedures analogous to those described in Example 91A.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US08119808B2uspto-grants-2012_02