Reaktion #1712989

ord-d487ca061b334b519fafc85cb9432921

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Aufarbeitung

  1. 1
    workup.ADDITIONwere treated in a manner similar to Reference Example 7
  2. 2
    Sonstigeto give the target compound

Vorschrift

5,7-Dimethylbenzo[b]thiophene (see Yoshimura, Y. et al., J. Med. Chem. 43 (2000) 2929-2937) and 5-bromo-2-chlorobenzaldehyde obtained in Reference Example 16-(1) were treated in a manner similar to Reference Example 7 to give the target compound.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US08785403B2uspto-grants-2014_07