Reaktion #168103

Reaktionsgleichung

1-(6-chloro-pyridazin-3-yl)-4-isopropyl-perhydro-1,4-diazepine

4-aminophenylboronic acid

pinacol cyclic ester

→

title compound

4-[6-(4-Isopropyl-perhydro-1,4-diazepin-1-yl)-pyridazin-3-yl]-phenylamine

Reaktionsbedingungen

Vorschrift

The title compound was prepared by a similar procedure to that described in Example 68, starting from 1-(6-chloro-pyridazin-3-yl)-4-isopropyl-perhydro-1,4-diazepine and 4-aminophenylboronic acid, pinacol cyclic ester. 1H NMR (400 MHz, CDCl3) δ 7.82 (d, 2H), 7.53 (d, 1H), 6.76 (m, 3H), 3.86 (t, 2H), 3.77 (m, 4H), 2.93 (heptet, 1H), 2.81 (m, 2H), 2.58 (m, 2H), 1.95 (m, 2H), 1.00 (d, 6H).

Quelle