Reaktion #160262

ord-8cc3981557c9491c93ba1f6a42bbe5fd

Reaktionsgleichung

COC(=O)c1ccc(S(=O)(=O)Cl)cc1
methyl 4-(chlorosulfonyl)benzoate
CCn1cc2cc(CN)ccc2n1
(2-ethyl-2H-indazol-5-yl)methanamine
→
CCn1cc2cc(CNS(=O)(=O)c3ccc(C(=O)OC)cc3)ccc2n1
titled compound
CCn1cc2cc(CNS(=O)(=O)c3ccc(C(=O)OC)cc3)ccc2n1
Methyl 4-(N-((2-ethyl-2H-indazol-5-yl)methyl)sulfamoyl)benzoate

Edukte

COC(=O)c1ccc(S(=O)(=O)Cl)cc1
methyl 4-(chlorosulfonyl)benzoate
CCn1cc2cc(CN)ccc2n1
(2-ethyl-2H-indazol-5-yl)methanamine

Reagenzien

Keine

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

The titled compound was prepared according to the procedure described in step-1 of Example 1 from methyl 4-(chlorosulfonyl)benzoate and (2-ethyl-2H-indazol-5-yl)methanamine (step-4 of Example 13).

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US08829026B2uspto-grants-2014_09