Reaktion #159687

Reaktionsgleichung

5-chloro-2-(3-(3-fluorophenyl)-3-hydroxyazetidin-1-yl)nicotinic acid

methyl 4-(1-aminocyclopropyl)benzoate hydrochloride

→

title compound ( D161 )

Ausbeute 66.9%

methyl 4-(1-(5-chloro-2-(3-(3-fluorophenyl)-3-hydroxyazetidin-1-yl)nicotinamido)cyclopropyl)benzoate

Ausbeute 66.9%

Reaktionsbedingungen

Aufarbeitung

1. 1
   Sonstigedescribed in Description 146 (reaction time 1 h)

Vorschrift

The title compound (D161) (64.7 mg) was prepared according to the experimental procedure described in Description 146 (reaction time 1 h) starting from 5-chloro-2-(3-(3-fluorophenyl)-3-hydroxyazetidin-1-yl)nicotinic acid (D111) (63 mg, 0.195 mmol) and methyl 4-(1-aminocyclopropyl)benzoate hydrochloride (D7) (44.4 mg, 0.195 mmol).

Quelle