Reaktion #1562

ord-08b8b8866d334d3cae4bec9581c21467

Reaktionsgleichung

Cn1c(=O)[nH]c(=O)n(-c2cc([N+](=O)[O-])c(F)cc2Cl)c1=O
1-(2-chloro-4-fluoro-5-nitrophenyl)-3-methyl-s-triazine-2,4,6(1H,3H,5H)-trione
[H][H]
hydrogen
CN1CN=CN(c2cc(N)c(F)cc2Cl)C1
title product
CN1CN=CN(c2cc(N)c(F)cc2Cl)C1
1-(5-Amino-2-chloro-4-fluorophenyl)-3-methyl-s-triazine

Lösungsmittel

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Aufarbeitung

  1. 1
    FiltrationThe reaction mixture is then filtered
  2. 2
    Einengenconcentrated in vacuo

Vorschrift

A mixture of 1-(2-chloro-4-fluoro-5-nitrophenyl)-3-methyl-s-triazine-2,4,6(1H,3H,5H)-trione (28.5 g, 0.09 mol) and 5% platinum on activated carbon (1 g) in ethyl acetate is hydrogenated at 55 psi until hydrogen uptake is complete. The reaction mixture is then filtered and concentrated in vacuo to give the title product as a white solid, mp 244°-245° C.

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US05726126uspto-grants-1998_03