Reaktion #155935

Reaktionsgleichung

4-(3-methylsulfanyl-1H-indazol-6-yl)-3,6-dihydro-2H-pyridine-1-carboxylic acid tert-butyl ester

4-methyl-phenyl boronic acid

→

title compound

3-Methylsulfanyl-6-(1,2,3,6-tetrahydro-pyridin-4-yl)-1-p-tolyl-1H-indazole

Reaktionsbedingungen

Aufarbeitung

1. 1
   Sonstigeto yield an intermediate, which
2. 2
   Sonstigeto remove the N-Boc

Vorschrift

The title compound was prepared as a white solid by coupling 4-(3-methylsulfanyl-1H-indazol-6-yl)-3,6-dihydro-2H-pyridine-1-carboxylic acid tert-butyl ester and 4-methyl-phenyl boronic acid to yield an intermediate, which was de-protected to remove the N-Boc.

Quelle