Reaktion #1053531

ord-1a91471e051347d0825f8883cf3a54bd

Reaktionsbedingungen

Detaillierte Bedingungen
See reaction.notes.procedure_details.

Vorschrift

In analogy to example 14.1, Trifluoro-methanesulfonic acid 3-(4-trifluoromethyl-phenyl)-benzo[d]isothiazol-6-yl ester and 2-[Ethyl-(1-ethynyl-cyclohexyl)-amino]-ethanol were converted to yield 2-(Ethyl-{1-[3-(4-trifluoromethyl-phenyl)-benzo[d]isothiazol-6-ylethynyl]-cydohexyl}-amino)-ethanol as brown oil, MS: 473.3 (MH+).

Quelle

DOI: 10.6084/m9.figshare.5104873.v1Patent: US06951879B2uspto-grants-2005_10