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Reaction #168806
N-(1-methyl-1H-pyrazol-3-yl)-6-({5-[3-(tetrahydro-2H-pyran-2-yloxy)propoxy]pyridin-2-yl}oxy)quinazoline-4-amine
Ausbeute 97.0%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168807
6-{[5-(2,2-diethoxyethoxy)pyridin-2-yl]oxy}-N-(1-methyl-1H-pyrazol-3-yl)quinazoline-4-amine
Ausbeute 65.0%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168813
6-[(5-{2-[ethyl(methyl)amino]ethoxy}pyridin-2-yl)oxy]-N-(1-methyl-1H-pyrazol-3-yl)quinazoline-4-amine
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168814
compound
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168815
6-({3-chloro-5-[2-(1,3-dioxolan-2-yl)ethoxy]pyridin-2-yl}oxy)-N-(1-methyl-1H-pyrazol-3-yl)quinazoline-4-amine
Ausbeute 73.0%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168817
5-chloro-6-({4-[(1-methyl-1H-pyrazol-3-yl)amino]quinazolin-6-yl}oxy)pyridin-3-ol
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168818
compound
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168819
6-({5-[(1-isopropylazetidin-3-yl)oxy]pyridin-2-yl}oxy)-N-(1-methyl-1H-pyrazol-3-yl)quinazoline-4-amine
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168820
6-({5-[(1-ethylazetidin-3-yl)oxy]-3-fluoropyridin-2-yl}oxy)-N-(1-methyl-1H-pyrazol-3-yl)quinazoline-4-amine
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168822
N-(1-methyl-1H-pyrazol-3-yl)-6-[(5-{[(2R)-2-(tetrahydro-2H-pyran-2-yloxy)propyl]oxy}pyridin-2-yl)oxy]quinazoline-4-amine
Ausbeute 75.1%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168823
compound
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168824
tert-butyl 3-({[6-({4-[(1-methyl-1H-pyrazol-3-yl)amino]quinazolin-6-yl}oxy)pyridin-3-yl]oxy}methyl)azetidine-1-carboxylate
Ausbeute 90.0%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168825
tert-butyl 2-(2-{[6-({4-[(1-methyl-1H-pyrazol-3-yl)amino]quinazolin-6-yl}oxy)pyridin-3-yl]oxy}ethyl)pyrrolidine-1-carboxylate
Ausbeute 90.9%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168844
compound
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168845
compound
Ausbeute 28.1%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168847
6-{[5-((1R)-2-{[tert-butyl(dimethyl)silyl]oxy}-1-methylethoxy)-3-chloropyridin-2-yl]oxy}-N-(1-methyl-1H-pyrazol-3-yl)quinazoline-4-amine
Ausbeute 33.1%DOI: 10.6084/m9.figshare.5104873.v1
Reaction #168848
compound
DOI: 10.6084/m9.figshare.5104873.v1
Reaction #182006
DOI: 10.1039/C8SC04228D
Reaction #262473
DOI: 10.1039/C8SC04228D
Reaction #291622
DOI: 10.1039/C8SC04228D
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