Ts2O

C=CCOC(=O)C(CN1C(=O)c2cccc(F)c2C1=O)C(C)=O
Reaction #10995
desired product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2006_08
C=C1Cn2c(=O)ccc3ncc(Cl)c1c32
Reaction #43403
3-Chloro-4-methylidene-4,5-dihydro-7H-pyrrolo[3,2,1-de]-1,5-naphthyridin-7-one
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CC(C)(C)Nc1nccc2cc(F)c(Cl)cc12
Reaction #73472
pure desired product ( 95 )
Ausbeute 4.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2013_09
COc1ccc(Cn2cc(-c3ccnc(NC(C)(C)C)c3)c(-c3cccc(N=C(c4ccccc4)c4ccccc4)c3)n2)cc1
Reaction #74115
title compound
Ausbeute 73.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2013_09
COc1ccc(Cn2cc(-c3ccnc(NC(C)(C)C)c3)c(-c3cccc([N+](=O)[O-])c3)n2)cc1
Reaction #74135
title compound
Ausbeute 75.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2013_09
O=C(C[C@H]1COC(=O)N1)OCc1ccccc1
Reaction #85651
(S)-benzyl 2-(2-oxooxazolidin-4-yl)acetate
Ausbeute 80.7%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_09
CC(C)(C)Nc1cc(OCCc2ccsc2)c(I)cn1
Reaction #171778
N-tert-butyl-5-iodo-4-(2-(thiophen-3-yl)ethoxy)pyridin-2-amine
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09
C=CCC1(C)CC(c2cncc(Cl)c2)C(c2ccc(Cl)cc2)N(C(CC)CO)C1=O
Reaction #180857
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)
COS(=O)(=O)c1ccc(C)cc1.Cc1cc(-c2ccccc2)nc2cc(-c3nc([C@H]4CC[C@H](CO)CC4)n4ccnc(N)c34)ccc12
Reaction #331335
product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_02
Cc1ccc(S(=O)(=O)OC[C@H]2C[C@H](n3cc(-c4ccc5ccc(-c6ccccc6)nc5c4)c4c(N)ncnc43)C2)cc1
Reaction #331342
desired product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_02
Cc1ccc(S(=O)(=O)OC[C@H]2C[C@@H](n3cc(I)c4c(N)ncnc43)C2)cc1
Reaction #331349
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_02
COC(=O)[C@H]1C[C@@H](OS(=O)(=O)c2ccc(C)cc2)C1
Reaction #331355
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_02
Cc1ccc(S(=O)(=O)OC[C@H]2C[C@@H](c3ncc4c(Cl)nccn43)C2)cc1
Reaction #331415
cis-3-(8-Chloroimidazo[1,5-a]pyrazin-3-yl)cyclobutylmethyl toluene-4-sulfonate
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_02
Cc1ccccc1S(=O)(=O)OC1=C(C(=O)OCc2ccccc2)N2C(=O)CC2C1
Reaction #334667
benzyl 3-toluenesulfonyloxy-1-azabicyclo[3.2.0]hept-2-en-7-one-2-carboxylate
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1987_11
Cc1ccc(S(=O)(=O)OC2=C(C(=O)OCc3ccccc3)N3C(=O)CC3C2)cc1
Reaction #334675
benzyl 3-(p-toluenesulfonyloxy)-1-azabicyclo[3.2.0]hept-2-en-7-one-2-carboxylate
Ausbeute 67.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1987_11
C=C1C[C@@H]2CC[C@@]34C[C@H]5O[C@H]6[C@@H](O3)[C@H]3O[C@H](CC[C@@H]3O[C@H]6[C@H]5O4)CC(=O)C[C@@H]3[C@@H](OC)[C@@H](C[C@H](O)CN)O[C@H]3C[C@H]3O[C@@H](CC[C@@H]1O2)C[C@@H](C)C3=C.CS(=O)(=O)O
Reaction #422707
B-1939
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_11
Cc1ccccc1S(=O)(=O)OC1=C(C(=O)OCc2ccccc2)N2C(=O)CC2C1
Reaction #458460
benzyl 3-toluenesulfonyloxy-1-azabicyclo[3.2.0]hept-2-en-7-one-2-carboxylate
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1985_07
Cc1ccc(S(=O)(=O)OC2=C(C(=O)OCc3ccccc3)N3C(=O)CC3C2)cc1
Reaction #458468
benzyl 3-(p-toluenesulfonyloxy)-1-azabicyclo[3.2.0]hept-2-en-7-one-2-carboxylate
Ausbeute 67.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1985_07
COS(=O)(=O)c1ccc(C)cc1.Cc1cc(-c2ccccc2)nc2cc(-c3nc([C@H]4CC[C@H](CO)CC4)n4ccnc(N)c34)ccc12
Reaction #473413
product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2013_02
Cc1ccc(S(=O)(=O)OC[C@H]2C[C@H](n3cc(-c4ccc5ccc(-c6ccccc6)nc5c4)c4c(N)ncnc43)C2)cc1
Reaction #473420
desired product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2013_02
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