تفاعل #985256

ord-24a34c2f2b9348b9894262d50538ecf8

معادلة التفاعل

O=[N+]([O-])c1ccc(/C=C/CCl)cc1
trans-4-Nitrocinnamyl chloride
Nc1ccccc1S
2-aminothiophenol
O=C([O-])[O-].[Na+].[Na+]
sodium carbonate
O=[N+]([O-])c1ccc(/C=C/c2nc3ccccc3s2)cc1
product 11
المردود 85.1%
O=[N+]([O-])c1ccc(/C=C/c2nc3ccccc3s2)cc1
Trans-2-(4-Nitrophenylethenyl)benzothiazole
المردود 85.1%

الكواشف

لا شيء

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

المعالجة

  1. 1
    ترشيحThe participate was collected by filtration under reduced pressure
  2. 2
    أخرىRecrystallization from methanol

الإجراء التجريبي

trans-4-Nitrocinnamyl chloride 10 (1.77 g, 9.5 mmol, 1.2 eq.) in DMF (20 ml) was added dropwise to a solution of 2-aminothiophenol 9 (1.0 g, 8.0 mmol) in DMF(15 ml) at room temperature. The reaction mixture was stirred at room temperature for overnight. The reaction mixture was poured into a solution of 10% sodium carbonate (100 ml). The participate was collected by filtration under reduced pressure. Recrystallization from methanol gave 1.92 g (85.1%) of the product 11.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07351401B2uspto-grants-2008_04