تفاعل #961

ord-1537debbdfcd4c9fb2d97af472b6fc7c

معادلة التفاعل

OCC1CCN(Cc2ccccc2)C1
(3RS)-1-benzyl-3-hydroxymethyl pyrrolidine
O=S(Cl)Cl
thionyl chloride
ClCC1CCN(Cc2ccccc2)C1
(3RS)-1-benzyl-3-chloromethyl pyrrolidine

الكواشف

لا شيء

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

المعالجة

  1. 1
    أخرىThe mixture was evaporated
  2. 2
    workup.DISSOLUTIONthe residue was dissolved in water

الإجراء التجريبي

To a refluxing solution of 15.3 g (0.08 mole) (3RS)-1-benzyl-3-hydroxymethyl pyrrolidine in 220 ml CHCl3 was slowly added a solution of 330 ml thionyl chloride in 60 ml CHCl3, and the reflux was continued for one hour. The mixture was evaporated and the residue was dissolved in water.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US05723444uspto-grants-1998_03