تفاعل #816386

ord-7edc6e62b38842c4962ead419202b6d3

معادلة التفاعل

[C-]#N.[K+]
KCN
O=C(Cl)c1ccccc1
benzoyl chloride
ClCCl.O
water methylene chloride
c1ccc2c(c1)ccc1ncccc12
benzo(f)chinolin
N#CC1C=Cc2c(ccc3ccccc23)N1C(=O)c1ccccc1
3-cyano-4-benzoyl-3,4-dihydrobenzo(f)chinoline

الكواشف

لا شيء

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

المعالجة

  1. 1
    أخرىThe organic phase was separated
  2. 2
    غسيلwashed with water, 5% hydrochloric acid, water, 5% NaOH solution
  3. 3
    تجفيفAfter drying over magnesium sulfate
  4. 4
    أخرىthe solution was evaporated to dryness

الإجراء التجريبي

648 μl (5.58 mmol) benzoyl chloride was added to a two phase system of water/methylene chloride over a period of two hours. These two layers contain 500 mg (2.79 mmol) of benzo(f)chinolin in the methylene chloride layer and 545 mg (8.37 mmol) KCN in water. Stirring was continued for 6 hours. The organic phase was separated and washed with water, 5% hydrochloric acid, water, 5% NaOH solution, and again with water. After drying over magnesium sulfate, the solution was evaporated to dryness.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07582295B2uspto-grants-2009_09