تفاعل #746925

ord-97f4d324d02c4d80b084fbac4c70776d

معادلة التفاعل

Cc1ccc(N)cc1Nc1ncc(-c2ccc(C#N)cc2)o1
4-[2-(5-Amino-2-methyl-phenylamino)-oxazol-5-yl]-benzonitrile
COc1cc(NC(C)=O)cc(OC)c1
N-(3,5-dimethoxyphenyl)-acetamide
CC(=O)Nc1cc(N)ccc1C
N-(5-amino-2-methyl-phenyl)-acetamide
COc1cc(Nc2ncc(-c3ccc(C#N)cc3)o2)cc(OC)c1
4-[2-(3,5-Dimethoxy-phenylamino)-oxazol-5-yl]-benzonitrile
المردود 85.0%

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

الإجراء التجريبي

The same procedure outlined above in the preparation of 4-[2-(5-Amino-2-methyl-phenylamino)-oxazol-5-yl]-benzonitrile was used. However N-(3,5-dimethoxyphenyl)-acetamide was used instead N-(5-amino-2-methyl-phenyl)-acetamide. Yield=85%.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US08080669B2uspto-grants-2011_12